RAD140 | B1211

RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that demonstrates excellent affinity for the androgen receptor (Ki = 7 nM). It displays potent anabolic effects in rodents and non-human primates and good bioavailability. It also demonstrates neuroprotective properties in hippocampal neurons of rat kainite model.

RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that demonstrates excellent affinity for the androgen receptor (Ki = 7 nM). It displays potent anabolic effects in rodents and non-human primates and good bioavailability. It also demonstrates neuroprotective properties in hippocampal neurons of rat kainite model.

B1211 | RAD140 DataSheet

Alternate Name/Synonyms: 2-​chloro-​4-​[[(1R,​2S)​-​1-​[5-​(4-​cyanophenyl)​-​1,​3,​4-​oxadiazol-​2-​yl]​-​2-​hydroxypropyl]​amino]​-​3-​methyl-benzonit

Appearance: White Solid

Formulation: N/A

CAS Number: 1182367-47-0

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₂₀H₁₆ClN₅O₂

Molecular Weight: 393.83

Cell-Permeable?: Yes

Purity: ≥98% by HPLC

Solubilities: DMSO(>3 mg/ml)

Handling: Protect from air and light

Country of Origin: USA

Tag Line: A potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM )

MDL Number:

PubChem CID: 44200882

SMILES: CC1=C(C=CC(=C1Cl)C#N)NC(C2=NN=C(O2)C3=CC=C(C=C3)C#N)C(C)O

InChi: InChI=1S/C20H16ClN5O2/c1-11-16(8-7-15(10-23)17(11)21)24-18(12(2)27)20-26-25-19(28-20)14-5-3-13(9-22)4-6-14/h3-8,12,18,24,27H,1-2H3/t12-,18+/m0/s1

InChi Key: XMBUPPIEVAFYHO-KPZWWZAWSA-N