RAF265 (CHIR-265) is a potent and selective inhibitor of C-Raf/B-Raf/B-Raf V600E (IC₅₀ of 3-60 nM); displays potent inhibition on VEGFR2 phosphorylation with EC₅₀ of 30 nM. RAF265 inhibits the growth...
CHIR99021 trihydrochloride is the hydrochloride salt of the potent and highly selective glycogen synthase kinase-3β (GSK-3β) inhibitor CHIR99021 (Cat. No. 1677).CHIR99021 trihydrochloride is the...