Tiplaxtinin | B1634

Tiplaxtinin(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 µM.

Tiplaxtinin(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 µM.

B1634 | Tiplaxtinin DataSheet

Alternate Name/Synonyms: Tiplaxtinin, PAI-039; PAI039; PAI 039; Tiplasinin; 2-[1-benzyl-5-[4-(trifluoromethoxy)phenyl]indol-3-yl]-2-oxoacetic acid

Appearance: Solid

Formulation: N/A

CAS Number: 393105-53-8

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₂₄H₁₆F₃NO₄

Molecular Weight: 439.38

Cell-Permeable?: Yes

Purity: >98%

Solubilities: DMSO

Handling: Protect from air and light

Country of Origin: USA

Tag Line: A plasminogen activator inhibitor-1 inhibitor

MDL Number: MFCD09475615

PubChem CID: 6450819

SMILES: C1=CC=C(C=C1)CN2C=C(C3=C2C=CC(=C3)C4=CC=C(C=C4)OC(F)(F)F)C(=O)C(=O)O

InChi: 1S/C24H16F3NO4/c25-24(26,27)32-18-9-6-16(7-10-18)17-8-11-21-19(12-17)20(22(29)23(30)31)14-28(21)13-15-4-2-1-3-5-15/h1-12,14H,13H2,(H,30,31)

InChi Key: ODXQFEWQSHNQNI-UHFFFAOYSA-N