Description
A potent aminopeptidase inhibitor (Ki = 0.001-90 mM); inhibits enkephalin metabolism and leukotriene A4 hydrolase. Displays antitumor and immunostimulant properties.
Bestatin is a potent aminopeptidase inhibitor (Ki = 0.001-90 mM); inhibits enkephalin metabolism and leukotriene A4 hydrolase.
Alternate Name/Synonyms: ([2S,3R]-3-Amino-2-hydroxy-4-phenylbutanoyl)-L-leucine; Ubenimex
Appearance: White solid
Formulation: N/A
CAS Number: 58970-76-6
Structure Available?: Yes
Peptide sequence: N/A
Salt Form: No
Molecular Formula: C₁₆H₂₄N₂O₄
Molecular Weight: 308.38
Cell-Permeable?: No
Purity: ≥99%
Solubilities: DMSO or MeOH
Handling: Protect from air and moisture
Country of Origin: USA
Tag Line: A potent aminopeptidase inhibitor
MDL Number: MFCD00083262
PubChem CID: 72172
SMILES: CC(C)CC(C(=O)O)NC(=O)C(C(CC1=CC=CC=C1)N)O
InChi: InChI=1S/C16H24N2O4/c1-10(2)8-13(16(21)22)18-15(20)14(19)12(17)9-11-6-4-3-5-7-11/h3-7,10,12-14,19H,8-9,17H2,1-2H3,(H,18,20)(H,21,22)/t12-,13+,14+/m1/s1
InChi Key: VGGGPCQERPFHOB-RDBSUJKOSA-N
Additional Information
Storage Condition: |
+4°C |
Shipping Condition: |
RT |
Shelf Life: |
24 months |