Bikinin | 2034

Cell-permeable. A highly specific inhibitor for the 7 Arabidopsis GSK-3 like kinase that activates brassinosteroid (BR) signaling downstream of the BR receptor. Bikinin directly binds the GSK3 BIN2 and acts as an ATP-competitive inhibitor. Furthermore, bikinin inhibits the activity of six other Arabidopsis GSK3s.

Bikininm is a highly specific inhibitor for the 7 Arabidopsis GSK-3 like kinase that activates brassinosteroid (BR) signaling downstream of the BR receptor. Bikinin directly binds the GSK3 BIN2 and acts as an ATP-competitive inhibitor. Furthermore, bikinin inhibits the activity of six other Arabidopsis GSK3s.

2034 | Bikinin DataSheet

Alternate Name/Synonyms: 4-((5-Bromo-2-pyridinyl)amino)-4-oxobutanoic acid; Arabidopsis GSK-3 Inhibitor

Appearance: White solid

Formulation: N/A

CAS Number: 188011-69-0

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₉H₉BrN₂O₃

Molecular Weight: 273.08

Cell-Permeable?: Yes

Purity: ≥95% by HPLC

Solubilities: DMSO ( 5 mg/ml)

Handling: Protect from air and light

Country of Origin: USA

Tag Line: A highly specific inhibitor for the 7 Arabidopsis GSK-3 like kinase

MDL Number: MFCD00116442

PubChem CID: 647833

SMILES: C1=CC(=NC=C1Br)NC(=O)CCC(=O)O

InChi: InChI=1S/C9H9BrN2O3/c10-6-1-2-7(11-5-6)12-8(13)3-4-9(14)15/h1-2,5H,3-4H2,(H,14,15)(H,11,12,13)

InChi Key: XFYYQDHEDOXWGA-UHFFFAOYSA-N