BX-517 | B1764

BX-517, also known as PDK1 inhibitor2, is a potent and selective PDK1 inhibitor that binds to the ATP binding pocket.

BX-517, also known as PDK1 inhibitor2, is a potent and selective PDK1 inhibitor that binds to the ATP binding pocket.

B1764 | BX-517 DataSheet

Alternate Name/Synonyms: BX-517; BX 517; BX517; PDK1 inhibitor2; (Z)-N-(3-(1-(1H-pyrrol-2-yl)ethylidene)-2-hydroxy-3H-indol-5-yl)carbamimidic acid; [(3Z)-2-oxo-3-[1-(1H-pyrrol-2-yl)ethylidene]-1H-indol-5-yl]urea

Appearance: Solid

Formulation: N/A

CAS Number: 850717-64-5

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₁₅H₁₄N₄O₂

Molecular Weight: 282.3

Cell-Permeable?: Yes

Purity: >98%

Solubilities: DMSO

Handling: Protect from air and light

Country of Origin: USA

Tag Line: A potent and selective PDK1 inhibitor

MDL Number: N/A

PubChem CID: 11161844

SMILES: CC(=C1C2=C(C=CC(=C2)NC(=O)N)NC1=O)C3=CC=CN3

InChi: InChI=1S/C15H14N4O2/c1-8(11-3-2-6-17-11)13-10-7-9(18-15(16)21)4-5-12(10)19-14(13)20/h2-7,17H,1H3,(H,19,20)(H3,16,18,21)/b13-8-

InChi Key: DFURSNCTQGJRRX-JYRVWZFOSA-N