CAY-10441 | B2353

CAY-10441 is a potent and selective IP (prostacyclin) receptor antagonist. It displays high affinity for IP receptors. CAY-10441 antagonizes the carbaprostacyclin-induced activation of human neuroblastoma adenylate cyclase, blocking cyclic AMP accumulation in a dose-dependent manner.

CAY-10441 is a potent and selective IP (prostacyclin) receptor antagonist. It displays high affinity for IP receptors. CAY-10441 antagonizes the carbaprostacyclin-induced activation of human neuroblastoma adenylate cyclase, blocking cyclic AMP accumulation in a dose-dependent manner.

B2353 | CAY-10441 DataSheet

Alternate Name/Synonyms: 4,5-dihydro-N-[4-[[4-(1-methylethoxy)phenyl]methyl]phenyl]-1H-imadazol-2-amine,RO-1138452,RO1138452

Appearance: Crystalline solid

Formulation:

CAS Number: 221529-58-4

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: N/A

Molecular Formula: C₁₉H₂₃N₃O

Molecular Weight: 309.4

Cell-Permeable?: TRUE

Purity: ≥98%

Solubilities: ~20 m g/ml (DMSO) in 0

Handling: Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.

Country of Origin: USA

Tag Line: A potent and selective IP (prostacyclin) receptor antagonist

MDL Number:

PubChem CID: 9839644

SMILES: CC(C)OC1=CC=C(C=C1)CC2=CC=C(C=C2)NC3=NCCN3

InChi: InChI=1S/C19H23N3O/c1-14(2)23-18-9-5-16(6-10-18)13-15-3-7-17(8-4-15)22-19-20-11-12-21-19/h3-10,14H,11-13H2,1-2H3,(H2,20,21,22)

InChi Key: GYYRMJMXXLJZAB-UHFFFAOYSA-N