VUF 8430 dihydrobromide | B2925

VUF 8430 is a high affinity agonist (pKi = 7.5) for the histamine H4 receptor (pEC₅₀= 7.3). It is a moderate affinity agonist for the H3 receptor and is inactive at H1 and H2 receptor.

VUF 8430 is a high affinity agonist (pKi = 7.5) for the histamine H4 receptor (pEC₅₀= 7.3). It is a moderate affinity agonist for the H3 receptor and is inactive at H1 and H2 receptor.

B2925 | VUF 8430 dihydrobromide DataSheet

Alternate Name/Synonyms: 2-guanidinoethyl carbamimidothioate dihydrobromide, 2-(2-guanidinoethyl)isothiourea dihydrobromide; Pseudourea, 2-(2-guanidinoethyl)-2-thio-, dihydrobromide

Appearance: Solid

Formulation:

CAS Number: 100130-32-3

Structure Available?: True

Peptide sequence:

Salt Form: True

Molecular Formula: C₄H₁₃Br₂N₅S

Molecular Weight: 323.05

Cell-Permeable?: True

Purity: 97%

Solubilities: 24 mg/ml in Water in 0, 30 mg/ml in in DMSO

Handling: Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.

Country of Origin: USA

Tag Line: A potent histamine H4 receptor agonist

MDL Number:

PubChem CID: 3063227

SMILES: C(CSC(=N)N)N=C(N)N.Br.Br

InChi: InChI=1S/C4H11N5S.2BrH/c5-3(6)9-1-2-10-4(7)8;;/h1-2H2,(H3,7,8)(H4,5,6,9);2*1H

InChi Key: GPWJSTKHQMIXCA-UHFFFAOYSA-N