BMS-779788 | B2602

BMS-779788 is a LXR partial agonist with IC₅₀ values of 68 nM for LXRα and 14 nM for LXRβ. BMS-779788 induces LXR target genes in blood in vivo with an EC₅₀ = 610 nM, a value similar to its in vitro blood gene induction potency.

BMS-779788 is a LXR partial agonist with IC₅₀ values of 68 nM for LXRα and 14 nM for LXRβ. BMS-779788 induces LXR target genes in blood in vivo with an EC₅₀ = 610 nM, a value similar to its in vitro blood gene induction potency.

B2602 | BMS-779788 DataSheet

Alternate Name/Synonyms: 2-(2-(2-(2-chlorophenyl)propan-2-yl)-1-(3'-(methylsulfonyl)-[1,1'-biphenyl]-4-yl)-1H-imidazol-4-yl)propan-2-ol, BMS 779788, EXEL04286652, XL652, BMS779788, EXEL-04286652, XL-652

Appearance: White to off-white solid

Formulation:

CAS Number: 918348-67-1

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₂₈H₂₉ClN₂O₃S

Molecular Weight: 509.06

Cell-Permeable?: True

Purity: ≥98% by HPLC

Solubilities: in DMSO

Handling: Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.

Country of Origin: USA

Tag Line: A potent partial LXR agonist

MDL Number:

PubChem CID: 59251511

SMILES: CC(C)(C1=CC=CC=C1Cl)C2=NC(=CN2C3=CC=C(C=C3)C4=CC(=CC=C4)S(=O)(=O)C)C(C)(C)O

InChi: InChI=1S/C28H29ClN2O3S/c1-27(2,23-11-6-7-12-24(2

InChi Key: JLPURTXCSILYLW-UHFFFAOYSA-N