BQR-695 | B2078

BQR-695 is a potent and selective PI4K inhibitor. Displays potency against both human PI4KIIIβ and Plasmodium falciparum asexual blood stages (IC₅₀ values of 90 nM and 71 nM, respectively). Antimalarial compound.

BQR-695 is a potent and selective PI4K inhibitor. Displays potency against both human PI4KIIIβ and Plasmodium falciparum asexual blood stages (IC₅₀ values of 90 nM and 71 nM, respectively). Antimalarial compound.

B2078 | BQR-695 DataSheet

Alternate Name/Synonyms: 2-((7-(3,4-dimethoxyphenyl)quinoxalin-2-yl)amino)-N-methylacetamide; NVP-BQR695

Appearance: Crystalline solid

Formulation: N/A

CAS Number: 1513879-21-4

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₁₉H₂₀Cl₂N₄O₃

Molecular Weight: 352.39

Cell-Permeable?: Yes

Purity: ≥98% by HPLC

Solubilities: DMSO

Handling: Protect from air and light

Country of Origin: USA

Tag Line: A potent and selective PI4K inhibitor

MDL Number: N/A

PubChem CID: 112499905

SMILES: CNC(=O)CNC1=CN=C2C=CC(=CC2=N1)C3=CC(=C(C=C3)OC)OC

InChi: InChI=1S/C19H20N4O3/c1-20-19(24)11-22-18-10-21-14-6-4-12(8-15(14)23-18)13-5-7-16(25-2)17(9-13)26-3/h4-10H,11H2,1-3H3,(H,20,24)(H,22,23)

InChi Key: LYPCULYCGFOIDA-UHFFFAOYSA-N