Description
BQR-695 is a potent and selective PI4K inhibitor. Displays potency against both human PI4KIIIβ and Plasmodium falciparum asexual blood stages (IC₅₀ values of 90 nM and 71 nM, respectively). Antimalarial compound.
BQR-695 is a potent and selective PI4K inhibitor. Displays potency against both human PI4KIIIβ and Plasmodium falciparum asexual blood stages (IC₅₀ values of 90 nM and 71 nM, respectively). Antimalarial compound.
Alternate Name/Synonyms: 2-((7-(3,4-dimethoxyphenyl)quinoxalin-2-yl)amino)-N-methylacetamide; NVP-BQR695
Appearance: Crystalline solid
Formulation: N/A
CAS Number: 1513879-21-4
Structure Available?: Yes
Peptide sequence: N/A
Salt Form: No
Molecular Formula: C₁₉H₂₀Cl₂N₄O₃
Molecular Weight: 352.39
Cell-Permeable?: Yes
Purity: ≥98% by HPLC
Solubilities: DMSO
Handling: Protect from air and light
Country of Origin: USA
Tag Line: A potent and selective PI4K inhibitor
MDL Number: N/A
PubChem CID: 112499905
SMILES: CNC(=O)CNC1=CN=C2C=CC(=CC2=N1)C3=CC(=C(C=C3)OC)OC
InChi: InChI=1S/C19H20N4O3/c1-20-19(24)11-22-18-10-21-14-6-4-12(8-15(14)23-18)13-5-7-16(25-2)17(9-13)26-3/h4-10H,11H2,1-3H3,(H,20,24)(H,22,23)
InChi Key: LYPCULYCGFOIDA-UHFFFAOYSA-N
Additional Information
Storage Condition: |
-20°C |
Shipping Condition: |
Gel Pack |
Shelf Life: |
36 months |