Description
CNX1351 is a potent and selective inhibitor of PI3Kα with IC50 value of 6.8 nM
CNX1351 is a potent and selective inhibitor of PI3Kα with IC50 value of 6.8 nM
Alternate Name/Synonyms: CNX-1351; CNX1351; CNX 1351; 1-(4-((2-(1H-indazol-4-yl)-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)piperazin-1-yl)-6-methylhept-5-ene-1,4-dione
Appearance: Solid
Formulation: N/A
CAS Number: 1276105-89-5
Structure Available?: Yes
Peptide sequence: N/A
Salt Form: No
Molecular Formula: C₃₀H₃₅N₇O₃S
Molecular Weight: 573.71
Cell-Permeable?: Yes
Purity: >98%
Solubilities: DMSO
Handling: Protect from air and light
Country of Origin: USA
Tag Line: A potent and selective PI3Kα inhibitor
MDL Number: N/A
PubChem CID: 58441401
SMILES: CC(=CC(=O)CCC(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6)C
InChi: InChI=1S/C30H35N7O3S/c1-20(2)16-21(38)6-7-27(39)36-10-8-35(9-11-36)19-22-17-26-28(41-22)30(37-12-14-40-15-13-37)33-29(32-26)23-4-3-5-25-24(23)18-31-34-25/h3-5,16-18H,6-15,19H2,1-2H3,(H,31,34)
InChi Key: DLNUPKDFXMWRFP-UHFFFAOYSA-N
Additional Information
Storage Condition: |
-20°C |
Shipping Condition: |
Gel Pack |
Shelf Life: |
36 months |