FAAH Inhibitor, PF-622 | 1928

Cell-permeable. A potent and irreversible FAAH (Fatty Acid Amide Hydrolase) inhibitor. Inhibits FAAH in a time-dependent manner by covalently modifying the enzyme's active site serine (IC₅₀ = 33 nM). It is highly selective for FAAH relative to other mammalian serine hydrolases.

FAAH Inhibitor, PF-622 is a potent and irreversible FAAH (Fatty Acid Amide Hydrolase) inhibitor. Inhibits FAAH in a time-dependent manner by covalently modifying the enzyme's active site serine (IC₅₀ = 33 nM). It is highly selective for FAAH relative to other mammalian serine hydrolases.

1928 | FAAH Inhibitor, PF-622 DataSheet

Alternate Name/Synonyms: N-Phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carboxamide

Appearance: White soild

Formulation: N/A

CAS Number: 898235-65-9

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₂₁H₂₂N₄O

Molecular Weight: 346.43

Cell-Permeable?: Yes

Purity: ≥98% by TLC

Solubilities: DMSO (~25 mg/ml) or Ethanol (~ 3 mg/ml)

Handling: Protect from light and air

Country of Origin: USA

Tag Line: A potent and irreversible FAAH (Fatty Acid Amide Hydrolase) inhibitor

MDL Number: N/A

PubChem CID: 11515763

SMILES: C1CN(CCN1CC2=NC3=CC=CC=C3C=C2)C(=O)NC4=CC=CC=C4

InChi: InChI=1S/C21H22N4O/c26-21(23-18-7-2-1-3-8-18)25-14-12-24(13-15-25)16-19-11-10-17-6-4-5-9-20(17)22-19/h1-11H,12-16H2,(H,23,26)

InChi Key: SNTCRRMCALVGNL-UHFFFAOYSA-N