Irsogladine maleate | B2187

Irsogladine maleate is a potent phosphodiesterase 4 (PDE4) inhibitor that displays gastroprotective properties. It facilitates gap junction intercellular communication through muscarinic acetylcholine receptor binding. It is a potent inhibitor of angiogenesis in wild-type and plasminogen activator-deficient mice.

Irsogladine maleate is a potent phosphodiesterase 4 (PDE4) inhibitor that displays gastroprotective properties. It facilitates gap junction intercellular communication through muscarinic acetylcholine receptor binding. It is a potent inhibitor of angiogenesis in wild-type and plasminogen activator-deficient mice.

B2187 | Irsogladine maleate DataSheet

Alternate Name/Synonyms: 6-(2,5-Dichlorophenyl)-1,3,5-triazine-2,4-diamine maleate

Appearance: White solid

Formulation: N/A

CAS Number: 84504-69-8

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₉H₇Cl₂N₅.C₄H₄O₄

Molecular Weight: 372.18

Cell-Permeable?: Yes

Purity: ≥98% by HPLC

Solubilities: DMSO (>30 mg/ml) or EtOH (>30 mg/ml)

Handling: Protect from air and light

Country of Origin: USA

Tag Line: A potent phosphodiesterase 4 (PDE4) inhibitor

MDL Number: MFCD00873566

PubChem CID: 5282435

SMILES: C1=CC(=C(C=C1Cl)C2=NC(=NC(=N2)N)N)Cl.C(=CC(=O)O)C(=O)O

InChi: InChI=1S/C9H7Cl2N5.C4H4O4/c10-4-1-2-6(11)5(3-4)7-14-8(12)16-9(13)15-7;5-3(6)1-2-4(7)8/h1-3H,(H4,12,13,14,15,16);1-2H,(H,5,6)(H,7,8)/b;2-1-

InChi Key: PJLVTVAIERNDEQ-BTJKTKAUSA-N