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PD-123319 ditrifluoroacetate | 9640
- SKU:
- 26-9640-GEN
- Availability:
- Usually shipped in 5 working days
Description
PD-123319 is a potent, selective, non-peptide angiotensin AT2 receptor antagonist (IC₅₀ values are 34 and 210 nM in rat adrenal tissue and brain respectively). It has been used to selectively examine the specific roles for AT1R and AT2R in hypertensive and other vascular research-related models.
PD-123319 is a potent, selective, non-peptide angiotensin AT2 receptor antagonist (IC₅₀ values are 34 and 210 nM in rat adrenal tissue and brain respectively). It has been used to selectively examine the specific roles for AT1R and AT2R in hypertensive and other vascular research-related models.
9640 | PD-123319 ditrifluoroacetate DataSheet
Alternate Name/Synonyms: 1-[[4-(Dimethylamino)-3-methylphenyl]methyl]-5-(diphenylacetyl)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridine-6-carboxylic acid ditrifluoroacetate
Appearance: Off-white solid
Formulation: N/A
CAS Number: 136676-91-0
Structure Available?: Yes
Peptide sequence: N/A
Salt Form: No
Molecular Formula: C₃₁H₃₂N₄O₃.2CF₃CO₂H
Molecular Weight: 736.67
Cell-Permeable?: Yes
Purity: ≥98% by HPLC
Solubilities: H₂O (>70 mg/ml)
Handling: Protect from air and light
Country of Origin: USA
Tag Line: A potent, selective, non-peptide angiotensin AT2 receptor antagonist
MDL Number: MFCD11046022
PubChem CID: N/A
SMILES: O=C(C1CC2=C(N=CN2CC3=CC=C(N(C)C)C(C)=C3)CN1C(C(C4=CC=CC=C4)C5=CC=CC=C5)=O)O.O=C(O)C(F)(F)F.O=C(O)C(F)(F)F
InChi: InChI=1S/C31H32N4O3.2C2HF3O2/c1-21-16-22(14-15-26(21)33(2)3)18-34-20-32-25-19-35(28(31(37)38)17-27(25)34)30(36)29(23-10-6-4-7-11-23)24-12-8-5-9-13-24;2*3-2(4,5)1(6)7/h4-16,20,28-29H,17-19H2,1-3H3,(H,37,38);2*(H,6,7)
InChi Key: GPKQIEZLHVGJQH-UHFFFAOYSA-N
Additional Information
Storage Condition: |
-20°C |
Shipping Condition: |
Gel Pack |
Shelf Life: |
36 months |