PD 150,606 | 1906

Cell-permeable. A selective, non-competitive Calpain inhibitor (Ki = 210 nM and 370 nM for Calpain-1 and Calpain-2, respectively). Interacts with the calcium-binding domain of calpain.

PD 150, 606 is a selective, non-competitive Calpain inhibitor (Ki = 210 nM and 370 nM for Calpain-1 and Calpain-2, respectively). Interacts with the calcium-binding domain of calpain.

1906 | PD 150,606 DataSheet

Alternate Name/Synonyms: 3-(4-Iodophenyl)-2-mercapto-(Z)-2-propenoic acid

Appearance: Off-white solid

Formulation: N/A

CAS Number: 179528-45-1

Structure Available?: Yes

Peptide sequence: N/A

Salt Form: No

Molecular Formula: C₉H₇IO₂S

Molecular Weight: 306.12

Cell-Permeable?: Yes

Purity: ≥98% by NMR

Solubilities: DMSO (10 mg/ml) or EtOH (1 mg/ml)

Handling: Protect from air and light

Country of Origin: USA

Tag Line: A selective, non-competitive Calpain inhibitor

MDL Number: MFCD00949076

PubChem CID: 9839500

SMILES: C1=CC(=CC=C1C=C(C(=O)O)S)I

InChi: InChI=1S/C9H7IO2S/c10-7-3-1-6(2-4-7)5-8(13)9(11)12/h1-5,13H,(H,11, 12)/b8-5-

InChi Key: DJCVSFWGKYHMKH-YVMONPNESA-N